Grant
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
Applicants
- Lundbeck (Denmark)
[NORA names: Lundbeck; Private Research; Denmark; Europe, EU; Nordic; OECD]
Abstract
The present invention provides compounds according to the following formula (I) which are inhibitors of the PDE1 enzyme and their use as medicaments, in particular for the treatment of neurodegenerative disorders and psychiatric disorders. The present invention also provides pharmaceutical compositions comprising compounds of the invention and methods of treating disorders using the compounds of the invention. (Automatic translation with Google Translate, without legal value)
Patent Family Records (8)
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGÅRD MORTEN, (...more)
2024, ES-2967489-T3
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2023, EP-3529250-B1
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
H Lundbeck AS, Lundbeck (Denmark) J. KELLER, L.K. Rasmussen, M. Langer Road, (...more)
2022, CN-109843884-B
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2020, US-10633382-B2
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2019, US-20190308968-A1
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2019, EP-3529250-A1
Imidazopyrazines ketone, PyrazolopyrimidinonecGMP and Pyrazolopyridine ketone as PDE1 inhibitor
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGAERD MORTEN, (...more)
2019, CN-109843884-A
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H LUNDBECK AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGÅRD MORTEN, (...more)
2018, WO-2018073251-A1