Application

IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS

Patent Number EP-3529250-A1

Publication Year 2019

Application Year 2017

Priority Year 2016

Jurisdiction EP

Status Granted

Inventors

KEHLER JAN RASMUSSEN LARS KYHN LANGGÅRD MORTEN JESSING MIKKEL VITAL PAULO JORGE VIEIRA JUHL KARSTEN

Applicants

  1. Lundbeck (Denmark)
  2. [NORA names: Lundbeck; Private Research; Denmark; Europe, EU; Nordic; OECD]

Abstract

The present invention provides compounds according to formula (I) below that are PDE1 enzyme inhibitors and their use as medicaments, in particular for the treatment of neurodegenerative disorders and psychiatric disorders. The present invention also provides pharmaceutical compositions comprising compounds of the invention and methods of treating disorders using the compounds of the invention.

Patent Family Records (8)

Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors  

H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGÅRD MORTEN, (...more)

2024, ES-2967489-T3

IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS  

H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)

2023, EP-3529250-B1

Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors  

H Lundbeck AS, Lundbeck (Denmark) J. KELLER, L.K. Rasmussen, M. Langer Road, (...more)

2022, CN-109843884-B

Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors  

H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)

2020, US-10633382-B2

IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS  

H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)

2019, US-20190308968-A1

IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS

H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)

2019, EP-3529250-A1

Imidazopyrazines ketone, PyrazolopyrimidinonecGMP and Pyrazolopyridine ketone as PDE1 inhibitor  

H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGAERD MORTEN, (...more)

2019, CN-109843884-A

IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS  

H LUNDBECK AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGÅRD MORTEN, (...more)

2018, WO-2018073251-A1

Data Provider: Digital Science