Grant
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
Applicants
- Lundbeck (Denmark)
[NORA names: Lundbeck; Private Research; Denmark; Europe, EU; Nordic; OECD]
Abstract
The present invention provides compounds according to the following formula (I) which are PDE1 enzyme inhibitors and their use as medicaments, in particular for the treatment of neurodegenerative and psychiatric disorders. The invention also provides pharmaceutical compositions comprising the compounds of the invention and methods of treating disorders using the compounds of the invention.
Patent Family Records (8)
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGÅRD MORTEN, (...more)
2024, ES-2967489-T3
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2023, EP-3529250-B1
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
H Lundbeck AS, Lundbeck (Denmark) J. KELLER, L.K. Rasmussen, M. Langer Road, (...more)
2022, CN-109843884-B
Imidazopyrazinones, pyrazolopyrimidinones and pyrazolopyridinones as PDE1 inhibitors
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2020, US-10633382-B2
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2019, US-20190308968-A1
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS KYHN, LANGGÅRD MORTEN, (...more)
2019, EP-3529250-A1
Imidazopyrazines ketone, PyrazolopyrimidinonecGMP and Pyrazolopyridine ketone as PDE1 inhibitor
H Lundbeck AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGAERD MORTEN, (...more)
2019, CN-109843884-A
IMIDAZOPYRAZINONES, PYRAZOLOPYRIMIDINONES AND PYRAZOLOPYRIDINONES AS PDE1 INHIBITORS
H LUNDBECK AS, Lundbeck (Denmark) KEHLER JAN, RASMUSSEN LARS, LANGGÅRD MORTEN, (...more)
2018, WO-2018073251-A1