Application

New hGH polymer prodrug

Patent Number JP-2022033787-A

Publication Year 2022

Application Year 2021

Priority Year 2014

Jurisdiction JP

Status Granted

Inventors

Thomas KURPIERS Anna SPLANEMANN JOACHIM ZETTLER HARALD RAU EVELYN EXNER STEEN JENSEN RASMUSSEN GRETHE NORSKOV TORBEN LESSMANN THOMAS WEGGE Alina HERMANN NINA SCHUBERT

Applicants

  1. Ascendis Pharma (Denmark)
  2. [NORA names: Ascendis Pharma; Private Research; Denmark; Europe, EU; Nordic; OECD]

Abstract

PROBLEM TO BE SOLVED: To provide pharmaceutical formulations for treating diseases that can be treated with human growth hormone (hGH), where the formulations keep the injection volume low to allow reliable administration of a drug in a manner convenient for a patient.

SOLUTION: The present invention provides a polymeric human growth hormone prodrug and dry, liquid and reconstituted pharmaceutical formulations comprising the prodrug. The present invention further provides their use as medicaments for treatment of diseases which can be treated with growth hormone, and methods of treatment. The present invention also relates to methods of application of such polymeric human growth hormone prodrug or pharmaceutical formulation.

SELECTED DRAWING: None

COPYRIGHT: (C)2022,JPO&INPIT

Patent Family Records (60)

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2024, IL-251906-B2

Novel polymeric hGH prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2024, AU-2024201227-A1

Novel polymeric hGH prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2024, AU-2020270494-B2

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, KR-20230152187-A

NOVEL POLYMERIC HGH PRODRUGS  

아센디스 파마 엔도크리놀로지 디비전 에이/에스 ВЕГГЕ Томас, ЙЕНСЕН Стеен, КУРПИРС Томас, (...more)

2023, KR-102608645-B1

Novel hGH polymer prodrugs  

Ascendis Pharma (Denmark), Ascendis Pharma AS Thomas KURPIERS, Anna SPLANEMANN, JOACHIM ZETTLER, (...more)

2023, JP-2023052300-A

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2023, IL-307773-A

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2023, IL-251906-B1

New HGH polymeric prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, ES-2947818-T3

New HGH polymeric prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, ES-2864415-T9

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, EP-4218823-A3

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, EP-4218823-A2

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, EP-3653227-B9

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2023, EP-3237014-B1

Hitherto UNKNOWN POLYMERS HGH PRODUCTS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, ZETTLER JOACHIM, ZETTLER, JOACHIM, (...more)

2023, DK-3653227-T5

New polymeric high prodrugs  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, ZETTLER JOACHIM, ZETTLER, JOACHIM, (...more)

2023, DK-3237014-T3

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMAN ANNA, ZETTLER JOACHIM, (...more)

2022, RS-61734-B2

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2022, PL-3653227-T6

Lonapegsomatropin  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2022, NO-2022014-I1

Lonapegsomatropin  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2022, NL-301172-I2

Lonapegsomatropin  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2022, NL-301172-I1

NOVEL POLYMERIC HGH PRODRUGS.  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S ZETTLER JOACHIM, ZETTLER, JOACHIM, WEGGE THOMAS, (...more)

2022, MX-2022009155-A

New hGH polymer prodrug

Ascendis Pharma (Denmark), Ascendis Pharma AS Thomas KURPIERS, Anna SPLANEMANN, JOACHIM ZETTLER, (...more)

2022, JP-2022033787-A

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2022, HR-P20210400-T4

NEW POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS

2022, FR-22C1029-I1

Lonapegsomatropin  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2022, FI-C20220017-I1

Novel polymeric HCh prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2022, ES-2864415-T7

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2022, EP-3653227-B3

Hitherto UNKNOWN POLYMERS HGH PRODUCTS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, ZETTLER JOACHIM, ZETTLER, JOACHIM, (...more)

2022, DK-3653227-T6

INNOVATIVE POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2022, CY-1123963-T1

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, SI-3653227-T1

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, SG-10202105511R-A

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMAN ANNA, ZETTLER JOACHIM, (...more)

2021, RS-61734-B1

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S

2021, PT-3653227-T

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, PL-3653227-T3

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, LT-3653227-T

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma (Denmark), Ascendis Pharma AS Thomas KURPIERS, Anna SPLANEMANN, JOACHIM ZETTLER, (...more)

2021, JP-2021020932-A

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, HU-E053855-T2

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, HR-P20210400-T1

New polymeric prodrugs of HCh.  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, ES-2864415-T3

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, EP-3653227-B1

Hitherto UNKNOWN POLYMERS HGH PRODUCTS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S KURPIERS THOMAS, ZETTLER JOACHIM, ZETTLER, JOACHIM, (...more)

2021, DK-3653227-T3

Novel polymeric hGH prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2021, AU-2015348633-C1

Novel Polymeric hGH Prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2020, US-20200390864-A1

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2020, US-10799563-B2

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2020, RU-2718664-C2

NOVEL POLYMERIC HGH PRODRUGS  

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2020, EP-3653227-A1

polymeric hgh prodrugs  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S Alina HERMANN, THOMAS WEGGE, TORBEN LESSMANN, (...more)

2020, BR-112017009798-A8

Novel polymeric hGH prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2020, AU-2020270494-A1

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2020, AU-2015348633-B2

NEW POLYMERIC hGH MEDICINES  

Асцендис Фарма Эндокринолоджи Дивижн А/С ВЕГГЕ Томас, ЙЕНСЕН Стеен, КУРПИРС Томас, (...more)

2018, RU-2017121203-A

Novel Polymeric hGH Prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2017, US-20170354716-A1

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2017, SG-11201703870U-A

NOVEL POLYMERIC HGH PRODRUGS.  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S JOACHIM ZETTLER, NINA SCHUBERT, Anna SPLANEMANN, (...more)

2017, MX-2017006113-A

NOVEL POLYMERIC HGH PRODRUGS  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2017, KR-20170084267-A

NOVEL POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2017, EP-3237014-A1

polymeric hgh prodrugs  

ASCENDIS PHARMA ENDOCRINOLOGY DIV A/S Alina HERMANN, THOMAS WEGGE, TORBEN LESSMANN, (...more)

2017, BR-112017009798-A2

Novel polymeric hGH prodrugs  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SCHUBERT NINA, ZETTLER JOACHIM, (...more)

2017, AU-2015348633-A1

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2016, WO-2016079114-A1

POLYMERIC HGH PRODRUGS  

Ascendis Pharma Endocrinology Division AS KURPIERS THOMAS, SPLANEMANN ANNA, SPLANEMANN, Anna, (...more)

2016, CA-2968282-A1

Data Provider: Digital Science