CRYSTALLINE FORMS OF A MONOACYLGLYCEROL LIPASE INHIBITOR

Patent Number: CA-3234430-A1

Publication Year: 2023

Application Year: 2022

Priority Year: 2021

Jurisdictions: CA

Status: Pending

Inventors:

ALLAN AMY ANDREW SAMUEL GEORGE ANDREW SAMUEL GEORGE ANDREW SAMUEL GEORGE S. G. Andrew VETTER THOMAS VETTER THOMAS BUZARD DANIEL J BUZARD DANIEL J BUZARD DANIEL J CINCOTTI ANTONIO CINCOTTI ANTONIO Daniel J. Buzad PATTERSON ADAM ROSS A. ALLEN ALLAN AMY ALLAN AMY ALLAN AMY PATTERSON ADAM ROSS ROSS PATTERSON ADAM VETTER THOMAS EDWARDS RICHARD JAMES EDWARDS RICHARD JAMES GANCEDO SUSANA DEL RIO GANCEDO SUSANA DEL RIO GANCEDO SUSANA DEL RIO S. D.R. Ganseido WIENER JOHN J M ALLAN AMY ANDREW SAMUEL GEORGE BUZARD DANIEL J. CINCOTTI ANTONIO EDWARDS RICHARD JAMES GANCEDO SUSANA DEL RIO GRICE CHERYL A. A. Sincotti ANDREW SAMUEL GEORGE CINCOTTI ANTONIO CINCOTTI ANTONIO CINCOTTI ANTONIO JUHL MARTIN JUHL MARTIN JUHL MARTIN LOPEZ DE DIEGO HEIDI PATTERSON ADAM ROSS VETTER THOMAS WIENER JOHN J. M. A R Paterson BUZARD DANIEL J LOPEZ DE DIEGO HEIDI LOPEZ DE DIEGO HEIDI PATTERSON ADAM ROSS PATTERSON ADAM ROSS PATTERSON ADAM ROSS CINCOTTI ANTONIO EDWARDS RICHARD JAMES EDWARDS RICHARD JAMES EDWARDS RICHARD JAMES GRICE CHERYL A GRICE CHERYL A R.J. EDWARDS EDWARDS RICHARD JAMES T. Vettel VETTER THOMAS VETTER THOMAS VETTER THOMAS WIENER JOHN J M WIENER JOHN J M BUZARD DANIEL J BUZARD DANIEL J GANCEDO SUSANA DEL RIO JUHL MARTIN JUHL MARTIN JUHL MARTIN M. Zur ALLAN AMY ALLAN AMY GRICE CHERYL A H. Lopez de Digo LOPEZ DE DIEGO HEIDI LOPEZ DE DIEGO HEIDI LOPEZ DE DIEGO HEIDI Cheryl A. Grace DEL RIO GANCEDO SUSANA DEL RIO GANCEDO SUSANA GRICE CHERYL A GRICE CHERYL A GRICE CHERYL A JUHL MARTIN ANDREW SAMUEL GEORGE ANDREW SAMUEL GEORGE LOPEZ DE DIEGO HEIDI WIENER JOHN J M WIENER JOHN J M WIENER JOHN J M WIENER JOHN J. M.

Applicants:

  1. Lundbeck (Denmark)
  2. [NORA names: Lundbeck; Private Research; Denmark; Europe, EU; Nordic; OECD]

Abstract

Described herein are new crystalline forms of the MAGL inhibitor 1-(1-(2-(pyrrolidin-1-yl)-4-(trifluoromethyl)b enzyl)-1,8-diazaspiro[4.5]decane-8-carbonyl)-1H-pyrazole-3-carboxylic acid, or a pharmaceutically acceptable salt thereof.

Patent Family Records (7)

CRYSTALLINE FORMS OF A MONOACYLGLYCEROL LIPASE INHIBITOR  

ALLAN AMY, ANDREW SAMUEL GEORGE, BUZARD DANIEL J, CINCOTTI ANTONIO, EDWARDS RICHARD JAMES, GANCEDO SUSANA DEL RIO, GRICE CHERYL A, H LUNDBECK AS, JUHL MARTIN, LOPEZ DE DIEGO HEIDI, Lundbeck (Denmark), PATTERSON ADAM ROSS, VETTER THOMAS, WIENER JOHN J M ALLAN AMY, PATTERSON ADAM ROSS, VETTER THOMAS, (...more)

2024, IL-311850-A

Crystalline forms of monoacylglycerol lipase inhibitors  

H Lundbeck AS, Lundbeck (Denmark) S. G. Andrew, Daniel J. Buzad, A. ALLEN, (...more)

2024, CN-118139863-A

CRYSTALLINE FORMS OF A MONOACYLGLYCEROL LIPASE INHIBITOR  

H Lundbeck AS, Lundbeck (Denmark) ANDREW SAMUEL GEORGE, BUZARD DANIEL J, ALLAN AMY, (...more)

2024, AU-2022382274-A1

CRYSTALLINE FORMS OF A MONOACYL GLYCEROL LIPASE INHIBITOR  

H LUNDBECK AS, Lundbeck (Denmark) VETTER THOMAS, CINCOTTI ANTONIO, ROSS PATTERSON ADAM, (...more)

2024, AR-127545-A1

CRYSTALLINE FORMS OF A MONOACYLGLYCEROL LIPASE INHIBITOR  

H LUNDBECK AS, Lundbeck (Denmark) ANDREW SAMUEL GEORGE, BUZARD DANIEL J, ALLAN AMY, (...more)

2023, WO-2023078868-A1

CRYSTALLINE FORMS OF A MAGL INHIBITOR  

H Lundbeck AS, Lundbeck (Denmark) VETTER THOMAS, CINCOTTI ANTONIO, PATTERSON ADAM ROSS, (...more)

2023, US-20230265095-A1

CRYSTALLINE FORMS OF A MONOACYLGLYCEROL LIPASE INHIBITOR

H Lundbeck AS, Lundbeck (Denmark) ANDREW SAMUEL GEORGE, BUZARD DANIEL J, ALLAN AMY, (...more)

2023, CA-3234430-A1

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