AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT

Patent Number: CA-2991805-A1

Publication Year: 2017

Application Year: 2016

Priority Year: 2015

Jurisdictions: CA

Status: Pending

Inventors:

BIRSHUITZER J ¨ 1 RGEN BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA Boshuizen, Julia JACOBSEN KIRSTINE JULIA BOSHUIZEN JULIA BOSHUIZEN JULIA BOSHUIZEN PARREN PAUL クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ DANIEL PEEPER DANIEL PEEPER DE JONG ROB DITZEL HENRIK J RN PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL Parren, Paul W H I 0000-0002-4365-3859 PAUL PARREN PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL SIMON VAN DIJKHUIZEN RADERSMA RIEMKE クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK J RN DITZEL HENRIK JOERN DITZEL HENRIK JOERN DITZEL HENRIK JORN DITZEL HENRIK JORN DITZEL HENRIK JORN HENRIK JORN DITZEL HENRIK JORN DITZEL PARREN PAUL PARREN PAUL PEEPER DANIEL クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ BOSHUIZEN JULIA DITZEL HENRIK J RN DITZEL HENRIK J RN PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PARREN PAUL PAUL PARREN PAUL PARREN クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER Breij, Esther C W ESTHER BREIJ JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE JACOBSEN KIRSTINE KRISTINE JACOBSEN KRISTINE JACOBSEN クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER BREIJ ESTHER ESTHER BREIJ ESTHER BREIJ KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE Koopman, Louise A 0000-0001-7648-9867 LOUISE KOOPMAN PEEPER DANIEL SATIJN DAVID クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ BREIJ ESTHER KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE KOOPMAN LOUISE LOUISE KOOPMAN LOUISE KOOPMAN SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID Satijn, David P E SATINKIN DMITRIY VERZIJL DENNIS クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ EDWARD VAN DEN BRINK KOOPMAN LOUISE SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID SATIJN DAVID VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DIJKHUIZEN RADERSMA RIEMKE クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ Dennis VERZIJL EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK SATIJN DAVID VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VAN DEN BRINK EDWARD VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS Verzijl, Dennis 0000-0002-7716-9838 WITZKY DIETER クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ BOSHUIZEN JULIA DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB Dennis VERZIJL Dennis VERZIJL ROB DE JONG VAN DEN BRINK EDWARD VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS VERZIJL DENNIS クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB DE JONG ROB JACOBSEN KIRSTINE Riemke VAN DIJKHUIZEN RADERSMA ROB DE JONG ROB DE JONG VAN DIJKHUIZEN RADASMA ROB VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VERZIJL DENNIS クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ DANIEL PEEPER DE JONG ROB KOOPMAN LOUISE PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL PEEPER DANIEL Peeper, Daniel Simon Riemke VAN DIJKHUIZEN RADERSMA Riemke VAN DIJKHUIZEN RADERSMA VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE VAN DIJKHUIZEN RADERSMA RIEMKE クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ クープマン ルイーズ

Applicants:

  1. Genmab (Denmark)
  2. [NORA names: Genmab; Private Research; Denmark; Europe, EU; Nordic; OECD]

Abstract

Antibody-drug conjugates (ADCs) binding to human AXL for therapeutic use, particularly for treatment of melanoma in combination with one or more MAPK pathway inhibitors such as, e.g., a BRAF inhibitor and/or a MEK inhibitor.

Patent Family Records (41)

AXL-specific antibody-drug conjugate for cancer treatment  

Genmab (Denmark), Genmab AS クープマン ルイーズ, クープマン ルイーズ, サテン デイビッド, (...more)

2024, JP-7428680-B2

AXL-specific antibody-drug conjugate for cancer treatment  

Genmab (Denmark), Genmab AS JULIA BOSHUIZEN, DANIEL PEEPER, HENRIK JORN DITZEL, (...more)

2024, JP-2024038480-A

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS JACOBSEN KIRSTINE, DITZEL HENRIK J RN, DITZEL HENRIK JØRN, (...more)

2024, AU-2022259847-B2

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2024, AU-2017206967-B2

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2023, US-20230321261-A1

AXL-specific antibody drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS BIRSHUITZER J ¨ 1 RGEN, PARREN PAUL, BREIJ ESTHER, (...more)

2023, CN-116617410-A

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS JULIA BOSHUIZEN, PAUL PARREN, ESTHER BREIJ, (...more)

2022, JP-2022037170-A

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATIONS FOR THE TREATMENT OF CANCER  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2022, CY-1123983-T1

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2022, AU-2022259847-A1

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2022, AU-2016292762-B2

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) PARREN PAUL, DE JONG ROB, PEEPER DANIEL, (...more)

2021, ME-03772-B

AXL-Specific Antibodies-Drug Conjugates for Cancer Treatment  

Genmab (Denmark), Genmab AS クープマン ルイーズ, クープマン ルイーズ, サテン デイビッド, (...more)

2021, JP-6892431-B2

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS JULIA BOSHUIZEN, DANIEL PEEPER, HENRIK JORN DITZEL, (...more)

2021, JP-2021138727-A

Axl-specific antibody-drug conjugates for cancer treatment  

GENMAB AS, Genmab (Denmark)

2021, IL-256790-B

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL SIMON, DITZEL HENRIK J RN, (...more)

2020, US-20200397913-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK JORN, (...more)

2020, SI-3319993-T1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, RS-60141-B1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark)

2020, PT-3319993-T

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, PL-3319993-T3

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, LT-3319993-T

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK JOERN, (...more)

2020, HU-E049072-T2

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, HR-P20200551-T1

AXL-Specific Antibody-Drug Conjugates for Cancer Treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, ES-2784685-T3

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, EP-3730520-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2020, EP-3319993-B1

AXL-SPECIFIC antibody-drug conjugates for cancer treatment  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, VAN DIJKHUIZEN RADERSMA RIEMKE, PARREN PAUL, (...more)

2020, DK-3319993-T3

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Antoni van Leeuwenhoek Hospital, Genmab (Denmark), Genmab AS, Stichting Het Nederlands Kanker Instituut Boshuizen, Julia, Parren, Paul W H I, Breij, Esther C W, (...more)

2019, US-20190022243-A1

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS クープマン ルイーズ, クープマン ルイーズ, サテン デイビッド, (...more)

2019, JP-2019509257-A

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2018, US-20180326084-A1

AXL-specific antibody-drug conjugates for cancer treatment  

GENMAB A, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK JOERN, (...more)

2018, KR-20180033523-A

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS クープマン ルイーズ, クープマン ルイーズ, サテン デイビッド, (...more)

2018, JP-2018525354-A

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2018, EP-3402822-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2018, EP-3319993-A1

AXL specific antibodies medicine conjugate use for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2018, CN-108884165-A

AXL specific antibodies-drug conjugate use for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK JORN, (...more)

2018, CN-108368171-A

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2018, AU-2017206967-A1

AXL-specific antibody-drug conjugates for cancer treatment  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2018, AU-2016292762-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2017, WO-2017121877-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

GENMAB AS, Genmab (Denmark) BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK J RN, (...more)

2017, WO-2017009258-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT  

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PARREN PAUL, BREIJ ESTHER, (...more)

2017, CA-3010887-A1

AXL-SPECIFIC ANTIBODY-DRUG CONJUGATES FOR CANCER TREATMENT

Genmab (Denmark), Genmab AS BOSHUIZEN JULIA, PEEPER DANIEL, DITZEL HENRIK JORN, (...more)

2017, CA-2991805-A1

Data Provider: Digital Science